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Cholesterol Absorption Inhibitors: Uses, Common Brands, and Safety Info

Cholesterol absorption inhibitors are drugs that lower cholesterol levels by reducing the absorption of dietary cholesterol in the body. They are used alongside lifestyle changes and other medications to manage high cholesterol. Common brands include Zetia and Welchol. These drugs are generally safe, but may cause gastrointestinal side effects. It is important to inform your doctor of other medications and conditions before starting this class of drugs. Regular follow-up visits and a healthy lifestyle are essential for effective cholesterol management.

Cholesterol Absorption Inhibitors

Cholesterol absorption inhibitors belong to a class of drugs used to lower cholesterol levels in the body. These medications work by reducing the absorption of dietary cholesterol in the small intestine, leading to decreased levels of LDL (low-density lipoprotein) cholesterol, often referred to as "bad" cholesterol. This class of drugs can be an effective addition to lifestyle modifications and other lipid-lowering treatments in managing high cholesterol.

Uses

Cholesterol absorption inhibitors are primarily indicated for the treatment of high cholesterol. They are often prescribed to patients who cannot tolerate statins or have not achieved their cholesterol goals with traditional statin therapy alone. These medications are typically prescribed alongside a low-cholesterol diet and exercise regimen to further lower LDL cholesterol levels in the body.

Common Brands

Two common drugs in the cholesterol absorption inhibitors class include ezetimibe and colesevelam. Ezetimibe, marketed under the brand name Zetia, is available as a tablet and is often used in combination with statins. Colesevelam, marketed as Welchol, is available in tablet or powder form and is mainly prescribed to lower LDL cholesterol levels.

Safety

Cholesterol absorption inhibitors are generally considered safe and well-tolerated. However, like all medications, they may have potential side effects. The most commonly reported side effects include gastrointestinal discomfort such as diarrhea, constipation, abdominal pain, and flatulence. These symptoms are usually mild and temporary. As with any other medication, it is important to inform your healthcare provider about any other medications, supplements, or medical conditions you have before starting cholesterol absorption inhibitors. Your doctor will assess possible drug interactions and determine if this class of drugs is suitable for you. It is worth noting that cholesterol absorption inhibitors alone may not sufficiently reduce cholesterol levels. Therefore, it is crucial to maintain a healthy lifestyle, including regular exercise, a balanced diet, and avoiding smoking and excessive alcohol consumption. Regular follow-up visits with your healthcare provider will also help monitor the effectiveness and safety of this medication. In conclusion, cholesterol absorption inhibitors are a class of drugs used for lowering cholesterol levels, primarily LDL cholesterol. They are commonly used as adjunct therapy to lifestyle modifications and other lipid-lowering drugs. Talk to your doctor to determine if cholesterol absorption inhibitors are a suitable option for managing your cholesterol.

List of Cholesterol Absorption Inhibitors